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Assay Detail

CHEMBL653865

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibitory concentration for anti-HIV activity against HIV-IIIB in CEM-SS cells
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type CEM-SS
Confidence 1 — Organism
Curated By Intermediate

Target

CEM-SS (CHEMBL614548)
Type CELL-LINE
Organism Homo sapiens

Publication

Antiviral oligo- and polyribonucleotides containing selected triazolo[2,3-a]purines.
Tutonda MG, Buckheit RW, Agrawal VK, Broom AD.
J Med Chem (1998) 41 : 4958 -4964
PubMed 9836613 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 6.92 8.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL107217 DITIOCARB SODIUM 2.0 1 8.82
CHEMBL3144270 1 7.10
CHEMBL3144269 1 6.00
CHEMBL3144271 1 5.77
CHEMBL3144268 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL107217 DITIOCARB SODIUM IC50 = 1.5 nM 8.82
CHEMBL3144270 IC50 = 80.0 nM 7.10
CHEMBL3144269 IC50 = 1000.0 nM 6.00
CHEMBL3144271 IC50 = 1700.0 nM 5.77
CHEMBL3144268 IC50 > 7000.0 nM -