Assay Detail
Functional
CHEMBL653983
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity in CHO cell lines
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Cricetulus griseus |
| Cell Type | CHO |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Defining the molecular requirements for the selective delivery of polyamine conjugates into cells containing active polyamine transporters.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 11 | 4.89 | 5.31 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3216621 | — | — | 1 | 5.31 |
| CHEMBL558390 | — | — | 1 | 5.12 |
| CHEMBL543610 | — | — | 1 | 5.02 |
| CHEMBL544167 | — | — | 1 | 5.02 |
| CHEMBL555288 | — | — | 1 | 4.95 |
| CHEMBL542751 | — | — | 1 | 4.81 |
| CHEMBL3216180 | — | — | 1 | 4.80 |
| CHEMBL558813 | — | — | 1 | 4.76 |
| CHEMBL540552 | — | — | 1 | 4.18 |
| CHEMBL540336 | — | — | 1 | - |
| CHEMBL542262 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3216621 | — | IC50 | = | 4900.0 | nM | 5.31 |
| CHEMBL558390 | — | IC50 | = | 7600.0 | nM | 5.12 |
| CHEMBL543610 | — | IC50 | = | 9500.0 | nM | 5.02 |
| CHEMBL544167 | — | IC50 | = | 9500.0 | nM | 5.02 |
| CHEMBL555288 | — | IC50 | = | 11200.0 | nM | 4.95 |
| CHEMBL542751 | — | IC50 | = | 15500.0 | nM | 4.81 |
| CHEMBL3216180 | — | IC50 | = | 15900.0 | nM | 4.80 |
| CHEMBL558813 | — | IC50 | = | 17400.0 | nM | 4.76 |
| CHEMBL540552 | — | IC50 | = | 66700.0 | nM | 4.18 |
| CHEMBL540336 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL542262 | — | IC50 | > | 1000000.0 | nM | - |