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Assay Detail

CHEMBL654534

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibition of [125I]RANTES association with CCR5 expressed in CHO cells at 100 nM
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Cell Type CHO
Confidence 1 — Organism
Curated By Intermediate

Target

CHO (CHEMBL613853)
Type CELL-LINE
Organism Cricetulus griseus

Publication

Inhibition of protein-protein association by small molecules: approaches and progress.
Toogood PL.
J Med Chem (2002) 45 : 1543 -1558
PubMed 11931608 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 8.85 8.85

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL41275 1 8.85

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL41275 IC50 = 1.4 nM 8.85