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Assay Detail

CHEMBL654640

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Compound was tested in vitro for inhibition of growth of cytotoxic CV-1 cell line
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type CV-1
Confidence 1 — Organism
Curated By Intermediate

Target

CV-1 (CHEMBL613507)
Type CELL-LINE
Organism Chlorocebus aethiops

Publication

Structure-activity of novel rhodacyanine dyes as antitumor agents.
Kawakami M, Koya K, Ukai T, Tatsuta N, Ikegawa A, Ogawa K, Shishido T, Chen LB.
J Med Chem (1998) 41 : 130 -142
PubMed 9438030 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 5.13 5.85

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL280643 1 5.85
CHEMBL413815 1 5.54
CHEMBL34783 1 5.06
CHEMBL33502 1 4.88
CHEMBL31074 1 4.83
CHEMBL33149 1 4.63

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL280643 IC50 = 1400.0 nM 5.85
CHEMBL413815 IC50 = 2900.0 nM 5.54
CHEMBL34783 IC50 = 8700.0 nM 5.06
CHEMBL33502 IC50 = 13200.0 nM 4.88
CHEMBL31074 IC50 = 14700.0 nM 4.83
CHEMBL33149 IC50 = 23600.0 nM 4.63