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Assay Detail

CHEMBL656304

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Concentration required to protect CEM cells against cytopathicity of HIV-1 by 50%
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type CCRF-CEM
Confidence 1 — Organism
Curated By Intermediate

Target

CCRF-CEM (CHEMBL382)
Type CELL-LINE
Organism Homo sapiens

Publication

Enhancing the aqueous solubility of d4T-based phosphoramidate prodrugs.
Siddiqui A, McGuigan C, Ballatore C, Srinivasan S, De Clercq E, Balzarini J.
Bioorg Med Chem Lett (2000) 10 : 381 -384
PubMed 10714505 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 7.12 7.12

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL107184 1 7.12

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL107184 EC50 = 75.0 nM 7.12