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Assay Detail

CHEMBL658303

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Agonistic activity on inositol phosphate production by intact transfected CHO cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Cricetulus griseus
Cell Type CHO
Confidence 1 — Organism
Curated By Intermediate

Target

CHO (CHEMBL613853)
Type CELL-LINE
Organism Cricetulus griseus

Publication

Synthesis and biological characterisation of [3H]BBL454, a new CCK2 selective radiolabelled agonist displaying original pharmacological properties.
Bellier B, Dugave C, Etivant F, Genet R, Gigoux V, Garbay C.
Bioorg Med Chem Lett (2004) 14 : 369 -372
PubMed 14698161 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 8.70 8.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL420161 1 8.70

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL420161 EC50 = 2.0 nM 8.70