Assay Detail
Binding
CHEMBL661386
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In vitro inhibition of crude dog red blood cell carbonic anhydrase
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Canis lupus familiaris |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
Sulfonylmethanesulfonamide inhibitors of carbonic anhydrase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.70 | 5.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL27601 | BENZENESULFONAMIDE | — | 1 | 5.70 |
| CHEMBL69291 | ETHANESULFONIC ACID AMIDE | — | 1 | - |
| CHEMBL305268 | METHANESULFONAMIDE | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL27601 | BENZENESULFONAMIDE | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL69291 | ETHANESULFONIC ACID AMIDE | IC50 | = | 1000000.0 | nM | - |
| CHEMBL305268 | METHANESULFONAMIDE | IC50 | = | 1000000.0 | nM | - |