Assay Detail
Binding
CHEMBL661901
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The compound was tested for its potency to inhibit human Cathepsin G
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Janus compounds: dual inhibitors of proteinases
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 5.72 | 5.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL147013 | — | — | 1 | 5.77 |
| CHEMBL422675 | — | — | 1 | 5.66 |
| CHEMBL150384 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL147013 | — | Ki | = | 1700.0 | nM | 5.77 |
| CHEMBL422675 | — | Ki | = | 2200.0 | nM | 5.66 |
| CHEMBL150384 | — | Ki | > | 1000000.0 | nM | - |