Assay Detail
Binding
CHEMBL662401
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Inhibitory activity against cholecystokinin type A receptor from rat pancreas binding assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Cholecystokinin receptor type A (CHEMBL2871) ↗| Type | SINGLE PROTEIN |
| Organism | Rattus norvegicus |
Publication
Analogs of CCK incorporating conformationally constrained replacements for Asp32.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 8.77 | 10.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL323521 | — | — | 1 | 10.30 |
| CHEMBL3143146 | — | — | 1 | 7.23 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL323521 | — | IC50 | = | 0.05 | nM | 10.30 |
| CHEMBL3143146 | — | IC50 | = | 59.0 | nM | 7.23 |