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Assay Detail

CHEMBL662690

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Compound was evaluated for the inhibition of Carbonic anhydrase (Non competitive)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 4 — Cell-line / Tissue
Curated By Autocuration

Target

Carbonic anhydrase (CHEMBL2095180)
Type PROTEIN FAMILY
Organism Homo sapiens

Publication

N-Substituted sulfonamide carbonic anhydrase inhibitors with topical effects on intraocular pressure.
Duffel MW, Ing IS, Segarra TM, Dixson JA, Barfknecht CF, Schoenwald RD.
J Med Chem (1986) 29 : 1488 -1494
PubMed 3735316 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 9.10 9.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL20 ACETAZOLAMIDE 4.0 1 9.10

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL20 ACETAZOLAMIDE Ki = 0.8 nM 9.10