Assay Detail
Binding
CHEMBL664929
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Inhibitory concentration against Dipeptidyl peptidase IV (DPP IV)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
A potent dipeptide inhibitor of dipeptidyl peptidase IV.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.17 | 5.24 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL37260 | — | — | 1 | 5.24 |
| CHEMBL290598 | — | — | 1 | 5.16 |
| CHEMBL432081 | — | — | 1 | 5.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL37260 | — | IC50 | = | 5700.0 | nM | 5.24 |
| CHEMBL290598 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL432081 | — | IC50 | = | 7900.0 | nM | 5.10 |