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Assay Detail

CHEMBL668393

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Binding
Evaluated for inhibition of dihydrofolate reductase (DHFR) from Lactobacillus casei
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Lacticaseibacillus casei
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Dihydrofolate reductase (CHEMBL2902)
Type SINGLE PROTEIN
Organism Lactobacillus casei

Publication

Synthesis and antifolate activity of 5-methyl-5,10-dideaza analogues of aminopterin and folic acid and an alternative synthesis of 5,10-dideazatetrahydrofolic acid, a potent inhibitor of glycinamide ribonucleotide formyltransferase.
Piper JR, McCaleb GS, Montgomery JA, Kisliuk RL, Gaumont Y, Thorndike J, Sirotnak FM.
J Med Chem (1988) 31 : 2164 -2169
PubMed 3184124 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 6.24 7.80

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL34259 METHOTREXATE 4.0 1 7.80
CHEMBL69016 1 7.64
CHEMBL66864 1 4.80
CHEMBL267890 1 4.72
CHEMBL66389 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL34259 METHOTREXATE IC50 = 16.0 nM 7.80
CHEMBL69016 IC50 = 23.0 nM 7.64
CHEMBL66864 IC50 = 16000.0 nM 4.80
CHEMBL267890 IC50 = 19000.0 nM 4.72
CHEMBL66389 IC50 > 100000.0 nM -