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Assay Detail

CHEMBL675875

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Ability to inhibit [3H]haloperidol binding to dopamine receptor in rat striatal homogenate
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Rattus norvegicus
Confidence 5 — Multiple protein complex / RNA
Curated By Autocuration

Target

Dopamine receptor (CHEMBL2093868)
Type PROTEIN FAMILY
Organism Rattus norvegicus

Publication

Examination of a series of 8-[3-[bis(4-fluorophenyl)amino]propyl]-1-aryl-1,3,8- triazaspiro[4.5]decan-4-ones as potential antipsychotic agents.
Wise LD, Pattison IC, Butler DE, DeWald HA, Lewis EP, Lobbestael SJ, Tecle H, Coughenour LL, Downs DA, Poschel BP.
J Med Chem (1985) 28 : 1811 -1817
PubMed 2866248 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 8.39 9.55

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL54 HALOPERIDOL 4.0 1 9.55
CHEMBL42 CLOZAPINE 4.0 1 7.22

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL54 HALOPERIDOL IC50 = 0.28 nM 9.55
CHEMBL42 CLOZAPINE IC50 = 60.0 nM 7.22