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Assay Detail

CHEMBL677377

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [3H]WIN-35428 binding to the dopamine transporter in rat caudate putamen tissue.
37
Total Activities
37
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Tissue Caudate-putamen
Confidence 8 — Homologous single protein target
Curated By Expert

Target

Sodium-dependent dopamine transporter (CHEMBL338)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

CoMFA study of novel phenyl ring-substituted 3alpha-(diphenylmethoxy)tropane analogues at the dopamine transporter.
Newman AH, Izenwasser S, Robarge MJ, Kline RH.
J Med Chem (1999) 42 : 3502 -3509
PubMed 10479283 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 37 7.04 7.93

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL317757 DIFLUOROBENZTROPINE 1 7.93
CHEMBL3084868 1 7.82
CHEMBL3084896 1 7.72
CHEMBL3084884 1 7.70
CHEMBL3084892 1 7.68
CHEMBL3084870 1 7.66
CHEMBL3084906 1 7.63
CHEMBL3084902 1 7.63
CHEMBL3084879 1 7.57
CHEMBL3084908 1 7.55
CHEMBL310310 1 7.52
CHEMBL3084894 1 7.51
CHEMBL3084883 1 7.49
CHEMBL3084905 1 7.42
CHEMBL3084882 1 7.42
CHEMBL3084909 1 7.32
CHEMBL3084869 1 7.30
CHEMBL3084907 1 7.16
CHEMBL3084880 1 7.11
CHEMBL3084903 1 7.11
CHEMBL3084887 1 7.05
CHEMBL3084897 1 7.04
CHEMBL1201203 BENZTROPINE 4.0 1 6.93
CHEMBL3084901 1 6.73
CHEMBL3084893 1 6.73
CHEMBL3084881 1 6.73
CHEMBL3084900 1 6.71
CHEMBL3084899 1 6.71
CHEMBL3084910 1 6.64
CHEMBL3084872 1 6.53

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL317757 DIFLUOROBENZTROPINE Ki = 11.8 nM 7.93
CHEMBL3084868 Ki = 15.2 nM 7.82
CHEMBL3084896 Ki = 18.9 nM 7.72
CHEMBL3084884 Ki = 20.0 nM 7.70
CHEMBL3084892 Ki = 21.1 nM 7.68
CHEMBL3084870 Ki = 22.0 nM 7.66
CHEMBL3084906 Ki = 23.3 nM 7.63
CHEMBL3084902 Ki = 23.4 nM 7.63
CHEMBL3084879 Ki = 27.0 nM 7.57
CHEMBL3084908 Ki = 27.9 nM 7.55
CHEMBL310310 Ki = 30.0 nM 7.52
CHEMBL3084894 Ki = 30.9 nM 7.51
CHEMBL3084883 Ki = 32.2 nM 7.49
CHEMBL3084905 Ki = 38.2 nM 7.42
CHEMBL3084882 Ki = 37.9 nM 7.42
CHEMBL3084909 Ki = 47.4 nM 7.32
CHEMBL3084869 Ki = 50.0 nM 7.30
CHEMBL3084907 Ki = 68.5 nM 7.16
CHEMBL3084880 Ki = 78.4 nM 7.11
CHEMBL3084903 Ki = 78.0 nM 7.11
CHEMBL3084887 Ki = 88.1 nM 7.05
CHEMBL3084897 Ki = 91.6 nM 7.04
CHEMBL1201203 BENZTROPINE Ki = 118.0 nM 6.93
CHEMBL3084901 Ki = 187.0 nM 6.73
CHEMBL3084893 Ki = 187.0 nM 6.73
CHEMBL3084881 Ki = 187.0 nM 6.73
CHEMBL3084900 Ki = 196.0 nM 6.71
CHEMBL3084899 Ki = 197.0 nM 6.71
CHEMBL3084910 Ki = 228.0 nM 6.64
CHEMBL3084872 Ki = 297.0 nM 6.53
CHEMBL3084878 Ki = 309.0 nM 6.51
CHEMBL3084888 Ki = 420.0 nM 6.38
CHEMBL3084898 Ki = 520.0 nM 6.28
CHEMBL3084873 Ki = 635.0 nM 6.20
CHEMBL3084891 AMINOBENZTROPINE Ki = 1840.0 nM 5.74
CHEMBL3084866 Ki = 1920.0 nM 5.72
CHEMBL3084867 Ki = 2000.0 nM 5.70