Assay Detail
Binding
CHEMBL678684
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Dissociation constant for Fibroblast growth factor 1
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Validation of molecular docking calculations involving FGF-1 and FGF-2.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 20 | 6.24 | 8.11 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2303816 | — | — | 1 | 8.11 |
| CHEMBL2303817 | — | — | 1 | 6.89 |
| CHEMBL2093120 | — | — | 1 | 6.27 |
| CHEMBL3144211 | — | — | 1 | 6.13 |
| CHEMBL2303818 | — | — | 1 | 5.94 |
| CHEMBL2029141 | — | — | 1 | 5.92 |
| CHEMBL2303819 | — | — | 1 | 4.43 |
| CHEMBL1160124 | — | — | 1 | - |
| CHEMBL1160119 | — | — | 1 | - |
| CHEMBL1160112 | — | — | 1 | - |
| CHEMBL1160111 | — | — | 1 | - |
| CHEMBL2303820 | — | — | 1 | - |
| CHEMBL421 | SULFASALAZINE | 4.0 | 1 | - |
| CHEMBL1160118 | — | — | 1 | - |
| CHEMBL2029142 | — | — | 1 | - |
| CHEMBL1160126 | — | — | 1 | - |
| CHEMBL1160117 | NAPHTHALENE TRISULFONATE | — | 1 | - |
| CHEMBL2303821 | — | — | 1 | - |
| CHEMBL1160122 | — | — | 1 | - |
| CHEMBL1160123 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2303816 | — | Kd | = | 7.8 | nM | 8.11 |
| CHEMBL2303817 | — | Kd | = | 130.0 | nM | 6.89 |
| CHEMBL2093120 | — | Kd | = | 540.0 | nM | 6.27 |
| CHEMBL3144211 | — | Kd | = | 740.0 | nM | 6.13 |
| CHEMBL2303818 | — | Kd | = | 1150.0 | nM | 5.94 |
| CHEMBL2029141 | — | Kd | = | 1200.0 | nM | 5.92 |
| CHEMBL2303819 | — | Kd | = | 37500.0 | nM | 4.43 |
| CHEMBL1160124 | — | Kd | = | 340000.0 | nM | - |
| CHEMBL1160119 | — | Kd | = | 337500.0 | nM | - |
| CHEMBL1160112 | — | Kd | = | 3410000.0 | nM | - |
| CHEMBL1160111 | — | Kd | = | 3250000.0 | nM | - |
| CHEMBL2303820 | — | Kd | = | 921000.0 | nM | - |
| CHEMBL421 | SULFASALAZINE | Kd | = | 609000.0 | nM | - |
| CHEMBL1160118 | — | Kd | = | 1340000.0 | nM | - |
| CHEMBL2029142 | — | Kd | = | 127000.0 | nM | - |
| CHEMBL1160126 | — | Kd | = | 120000.0 | nM | - |
| CHEMBL1160117 | NAPHTHALENE TRISULFONATE | Kd | = | 474000.0 | nM | - |
| CHEMBL2303821 | — | Kd | = | 300000.0 | nM | - |
| CHEMBL1160122 | — | Kd | = | 307000.0 | nM | - |
| CHEMBL1160123 | — | Kd | = | 5940000.0 | nM | - |