Assay Detail
Binding
CHEMBL681265
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of Fucosyltransferase 5 by the compound was evaluated; Competitive inhibition
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5 (CHEMBL3146) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Inhibition kinetics of carba- and C-fucosyl analogues of GDP-fucose against fucosyltransferase V: implication for the reaction mechanism.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 4.17 | 4.17 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL609638 | — | — | 1 | 4.17 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL609638 | — | Ki | = | 67100.0 | nM | 4.17 |