Assay Detail
Binding
CHEMBL681649
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of yeast Farnesyl transferase
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Saccharomyces cerevisiae |
| Confidence | 6 — Multiple protein complex / RNA |
| Curated By | Expert |
Target
Farnesyltransferase (CHEMBL2111393) ↗| Type | PROTEIN COMPLEX |
| Organism | Saccharomyces cerevisiae S288c |
Publication
Synthesis and evaluation of benzophenone-based photoaffinity labeling analogs of prenyl pyrophosphates containing stable amide linkages
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 7.12 | 7.12 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL69330 | FARNESYL DIPHOSPHATE | — | 1 | 7.12 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL69330 | FARNESYL DIPHOSPHATE | Kd | = | 75.0 | nM | 7.12 |