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Assay Detail

CHEMBL681671

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Binding
Inhibitory activity against the human recombinant geranylgeranyl diphosphate synthase (GGPPSase).
29
Total Activities
29
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Expert

Target

Geranylgeranyl pyrophosphate synthase (CHEMBL4769)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Inhibition of geranylgeranyl diphosphate synthase by bisphosphonates and diphosphates: a potential route to new bone antiresorption and antiparasitic agents.
Szabo CM, Matsumura Y, Fukura S, Martin MB, Sanders JM, Sengupta S, Cieslak JA, Loftus TC, Lea CR, Lee HJ, Koohang A, Coates RM, Sagami H, Oldfield E.
J Med Chem (2002) 45 : 2185 -2196
PubMed 12014956 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 29 5.62 6.85

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL71360 1 6.85
CHEMBL419627 1 6.51
CHEMBL67986 1 6.43
CHEMBL54004 1 6.14
CHEMBL71017 1 6.13
CHEMBL416301 1 6.04
CHEMBL298852 1 5.85
CHEMBL52251 (OCTYLAMINO)METHYLENEDIPHOSPHONIC ACID 1 5.66
CHEMBL298547 1 5.37
CHEMBL55264 1 4.96
CHEMBL56254 (HEXYLAMINO)METHYLENEDIPHOSPHONIC ACID 1 4.72
CHEMBL299988 1 4.28
CHEMBL997 IBANDRONIC ACID 4.0 1 4.08
CHEMBL305530 1 -
CHEMBL299491 1 -
CHEMBL55557 1 -
CHEMBL68666 1 -
CHEMBL56556 1 -
CHEMBL55358 1 -
CHEMBL417932 1 -
CHEMBL52761 1 -
CHEMBL55214 NERIDRONIC ACID 3.0 1 -
CHEMBL301247 1 -
CHEMBL870 ALENDRONIC ACID 4.0 1 -
CHEMBL834 PAMIDRONIC ACID 4.0 1 -
CHEMBL923 RISEDRONIC ACID 4.0 1 -
CHEMBL293522 1 -
CHEMBL55140 1 -
CHEMBL55359 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL71360 IC50 = 140.0 nM 6.85
CHEMBL419627 IC50 = 310.0 nM 6.51
CHEMBL67986 IC50 = 370.0 nM 6.43
CHEMBL54004 IC50 = 720.0 nM 6.14
CHEMBL71017 IC50 = 740.0 nM 6.13
CHEMBL416301 IC50 = 920.0 nM 6.04
CHEMBL298852 IC50 = 1400.0 nM 5.85
CHEMBL52251 (OCTYLAMINO)METHYLENEDIPHOSPHONIC ACID IC50 = 2200.0 nM 5.66
CHEMBL298547 IC50 = 4300.0 nM 5.37
CHEMBL55264 IC50 = 11000.0 nM 4.96
CHEMBL56254 (HEXYLAMINO)METHYLENEDIPHOSPHONIC ACID IC50 = 19000.0 nM 4.72
CHEMBL299988 IC50 = 53000.0 nM 4.28
CHEMBL997 IBANDRONIC ACID IC50 = 83000.0 nM 4.08
CHEMBL305530 IC50 > 100000.0 nM -
CHEMBL299491 IC50 = 200000.0 nM -
CHEMBL55557 IC50 = 260000.0 nM -
CHEMBL68666 IC50 = 240000.0 nM -
CHEMBL56556 IC50 = 220000.0 nM -
CHEMBL55358 IC50 = 330000.0 nM -
CHEMBL417932 IC50 = 180000.0 nM -
CHEMBL52761 IC50 = 620000.0 nM -
CHEMBL55214 NERIDRONIC ACID IC50 = 690000.0 nM -
CHEMBL301247 IC50 = 220000.0 nM -
CHEMBL870 ALENDRONIC ACID IC50 = 440000.0 nM -
CHEMBL834 PAMIDRONIC ACID IC50 = 180000.0 nM -
CHEMBL923 RISEDRONIC ACID IC50 = 350000.0 nM -
CHEMBL293522 IC50 = 410000.0 nM -
CHEMBL55140 IC50 = 220000.0 nM -
CHEMBL55359 IC50 = 550000.0 nM -