Assay Detail
Binding
CHEMBL681696
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Compound was evaluated for its ability to displace radiolabeled glucagon
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Development of potent truncated glucagon antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.88 | 8.43 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL413890 | — | — | 1 | 8.43 |
| CHEMBL438045 | — | — | 1 | 7.32 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL413890 | — | IC50 | = | 3.75 | nM | 8.43 |
| CHEMBL438045 | — | IC50 | = | 48.0 | nM | 7.32 |