Glucagon receptor · SINGLE PROTEIN · Rattus norvegicus
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As of 2026-09-14Protein identity stays anchored to UniProt P30082. Use UniProt P30082 as the stable identity anchor, then attach disease evidence before program review.
Use UniProt P30082 as the stable identity anchor, then attach disease evidence before program review.
Glucagon receptor
Review this target as Glucagon receptor, mapped to UniProt P30082. Sequence length is 485 aa.
Protein source · UniProt accession via ChEMBL component mappingKeep the review anchor, source IDs, and context contract aligned before reusing this target elsewhere.
This review treats Glucagon receptor as ChEMBL target CHEMBL4720, mapped to UniProt P30082. Disease framing currently uses the Open Targets-ready proxy contract.
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Start here when your first question is whether Glucagon receptor is the right protein anchor across sources, using UniProt P30082 as the stable mapping.
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| Preferred Name | Glucagon receptor |
| Target Type | SINGLE PROTEIN |
| Organism | Rattus norvegicus |
| UniProt | P30082 |
Reviewable protein naming and mapping context for this target snapshot.
| Protein Label | Glucagon receptor |
| UniProt Accession | P30082 |
| Component Type | Protein |
| Sequence Length | 485 aa |
Glucagon receptor
Review this target as Glucagon receptor, mapped to UniProt P30082. Sequence length is 485 aa.
| ChEMBL ID | pChEMBL | Type | Value (nM) | Phase |
|---|---|---|---|---|
| CHEMBL428460 | 9.7 | IC50 | 0.2 | Preclinical |
| CHEMBL412488 | 9.62 | IC50 | 0.24 | Preclinical |
| CHEMBL152640 | 9.37 | IC50 | 0.43 | Preclinical |
| CHEMBL152765 | 9.0 | IC50 | 1.0 | Preclinical |
| CHEMBL429362 | 8.82 | IC50 | 1.5 | Preclinical |
| CHEMBL439885 | 8.77 | IC50 | 1.7 | Preclinical |
| CHEMBL413666 | 8.64 | IC50 | 2.3 | Preclinical |
| CHEMBL267189 | 8.44 | IC50 | 3.6 | Preclinical |
| CHEMBL413890 | 8.43 | IC50 | 3.75 | Preclinical |
| CHEMBL2115191 | 8.39 | IC50 | 4.1 | Preclinical |
| BAO Format | Assays | Compounds | Avg pChEMBL |
|---|---|---|---|
| single protein format | 24 | 53 | 7.2 |
| cell membrane format | 7 | 45 | 6.0 |
| assay format | 4 | 7 | 6.4 |
| tissue-based format | 1 | 2 | 6.2 |
| BAO Format | Assays | Compounds | Avg pChEMBL |
|---|---|---|---|
| cell-based format | 8 | 3 | 7.3 |
| assay format | 2 | 1 | 5.6 |