Assay Detail
Binding
CHEMBL682012
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Inhibitory activity against Rabbit factor Xa was determined
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Oryctolagus cuniculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Intermediate |
Publication
Nonbenzamidine isoxazoline derivatives as factor Xa inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 8.98 | 9.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL7651 | — | — | 1 | 9.96 |
| CHEMBL7626 | — | — | 1 | 8.64 |
| CHEMBL267438 | — | — | 1 | 8.33 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL7651 | — | Ki | = | 0.11 | nM | 9.96 |
| CHEMBL7626 | — | Ki | = | 2.3 | nM | 8.64 |
| CHEMBL267438 | — | Ki | = | 4.7 | nM | 8.33 |