Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL682022

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Tested for inhibitory activity against Coagulation factor Xa
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Coagulation factor X (CHEMBL244)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Benzimidazoles and isosteric compounds as potent and selective factor Xa inhibitors.
He W, Hanney B, Myers MR, Condon S, Becker MR, Spada AP, Burns C, Brown K, Colussi D, Chu V.
Bioorg Med Chem Lett (2002) 12 : 919 -922
PubMed 11958994 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 7.38 7.38

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL354996 1 7.38

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL354996 Ki = 42.0 nM 7.38