Assay Detail
Functional
CHEMBL691178
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Effective dose measuring intracellular calcium elevation in HEK293 cells
27
Total Activities
27
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 1 — Organism |
| Curated By | Expert |
Publication
Structure-function studies on the new growth hormone-releasing peptide, ghrelin: minimal sequence of ghrelin necessary for activation of growth hormone secretagogue receptor 1a.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 27 | 7.23 | 8.08 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL526723 | — | — | 1 | 8.08 |
| CHEMBL2310891 | — | — | 1 | 8.04 |
| CHEMBL422461 | — | — | 1 | 7.94 |
| CHEMBL2310888 | — | — | 1 | 7.82 |
| CHEMBL410108 | — | — | 1 | 7.77 |
| CHEMBL501253 | — | — | 1 | 7.75 |
| CHEMBL263544 | — | — | 1 | 7.70 |
| CHEMBL412799 | — | — | 1 | 7.66 |
| CHEMBL525994 | — | — | 1 | 7.62 |
| CHEMBL504776 | — | — | 1 | 7.51 |
| CHEMBL425281 | — | — | 1 | 7.50 |
| CHEMBL2310887 | — | — | 1 | 7.42 |
| CHEMBL412565 | — | — | 1 | 7.42 |
| CHEMBL2310890 | — | — | 1 | 7.41 |
| CHEMBL2310893 | — | — | 1 | 7.38 |
| CHEMBL2310894 | — | — | 1 | 7.28 |
| CHEMBL335799 | — | — | 1 | 7.14 |
| CHEMBL2310886 | — | — | 1 | 6.39 |
| CHEMBL136092 | — | — | 1 | 5.94 |
| CHEMBL509512 | — | — | 1 | 5.92 |
| CHEMBL504856 | — | — | 1 | 5.70 |
| CHEMBL422630 | — | — | 1 | 5.60 |
| CHEMBL434649 | — | — | 1 | - |
| CHEMBL428282 | — | — | 1 | - |
| CHEMBL139427 | — | — | 1 | - |
| CHEMBL2310889 | — | — | 1 | - |
| CHEMBL2310892 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL526723 | — | EC50 | = | 8.3 | nM | 8.08 |
| CHEMBL2310891 | — | EC50 | = | 9.1 | nM | 8.04 |
| CHEMBL422461 | — | EC50 | = | 11.5 | nM | 7.94 |
| CHEMBL2310888 | — | EC50 | = | 15.0 | nM | 7.82 |
| CHEMBL410108 | — | EC50 | = | 17.0 | nM | 7.77 |
| CHEMBL501253 | — | EC50 | = | 18.0 | nM | 7.75 |
| CHEMBL263544 | — | EC50 | = | 20.0 | nM | 7.70 |
| CHEMBL412799 | — | EC50 | = | 22.0 | nM | 7.66 |
| CHEMBL525994 | — | EC50 | = | 24.0 | nM | 7.62 |
| CHEMBL504776 | — | EC50 | = | 31.0 | nM | 7.51 |
| CHEMBL425281 | — | EC50 | = | 32.0 | nM | 7.50 |
| CHEMBL2310887 | — | EC50 | = | 38.0 | nM | 7.42 |
| CHEMBL412565 | — | EC50 | = | 38.0 | nM | 7.42 |
| CHEMBL2310890 | — | EC50 | = | 39.0 | nM | 7.41 |
| CHEMBL2310893 | — | EC50 | = | 42.0 | nM | 7.38 |
| CHEMBL2310894 | — | EC50 | = | 53.0 | nM | 7.28 |
| CHEMBL335799 | — | EC50 | = | 72.0 | nM | 7.14 |
| CHEMBL2310886 | — | EC50 | = | 410.0 | nM | 6.39 |
| CHEMBL136092 | — | EC50 | = | 1150.0 | nM | 5.94 |
| CHEMBL509512 | — | EC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL504856 | — | EC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL422630 | — | EC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL434649 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL428282 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL139427 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL2310889 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL2310892 | — | EC50 | > | 10000.0 | nM | - |