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Assay Detail

CHEMBL691357

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibitory activity against HCMV DNA synthesis in virus infected cells
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HEL
Confidence 1 — Organism
Curated By Intermediate

Target

HEL (CHEMBL613888)
Type CELL-LINE
Organism Homo sapiens

Publication

Haloanilino derivatives of pyrimidines, purines, and purine nucleoside analogs: synthesis and activity against human cytomegalovirus.
Medveczky M, Yang TF, Gambino J, Medveczky P, Wright GE.
J Med Chem (1995) 38 : 1811 -1819
PubMed 7752205 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 8 4.74 5.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL51501 1 5.30
CHEMBL53912 1 5.04
CHEMBL51613 1 4.92
CHEMBL298714 1 4.60
CHEMBL54127 1 4.60
CHEMBL301283 1 4.55
CHEMBL53307 1 4.48
CHEMBL52034 1 4.40

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL51501 IC50 = 5000.0 nM 5.30
CHEMBL53912 IC50 = 9100.0 nM 5.04
CHEMBL51613 IC50 = 12000.0 nM 4.92
CHEMBL298714 IC50 = 25000.0 nM 4.60
CHEMBL54127 IC50 = 25000.0 nM 4.60
CHEMBL301283 IC50 = 28000.0 nM 4.55
CHEMBL53307 IC50 = 33000.0 nM 4.48
CHEMBL52034 IC50 = 40000.0 nM 4.40