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Assay Detail

CHEMBL694508

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Concentration required to reduce human cytomegalo virus(Davis) inducted cytopathicity by 50% (HEL cells)
8
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HEL
Confidence 1 — Organism
Curated By Intermediate

Target

HEL (CHEMBL613888)
Type CELL-LINE
Organism Homo sapiens

Publication

Polyanion inhibitors of human immunodeficiency virus and other viruses. 6. Micelle-like anti-HIV polyanionic compounds based on a carbohydrate core.
Leydet A, Jeantet-Segonds C, Bouchitté C, Moullet C, Boyer B, Roque JP, Witvrouw M, Este J, Snoeck R, Andrei G, De Clercq E.
J Med Chem (1997) 40 : 350 -356
PubMed 9022801 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 8 5.92 6.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3215377 1 6.40
CHEMBL3217279 1 5.44
CHEMBL3142956 1 -
CHEMBL384019 2 -
CHEMBL3215376 1 -
CHEMBL3142950 1 -
CHEMBL3215375 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3215377 IC50 = 400.0 nM 6.40
CHEMBL3217279 IC50 = 3600.0 nM 5.44
CHEMBL3142956 IC50 > 25000.0 nM -
CHEMBL384019 IC50 > 22000.0 nM -
CHEMBL3215376 IC50 > 333000.0 nM -
CHEMBL384019 IC50 > 22000.0 nM -
CHEMBL3142950 IC50 > 22000.0 nM -
CHEMBL3215375 IC50 > 37000.0 nM -