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Assay Detail

CHEMBL694727

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human foreskin fibroblasts (HFF) cells
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HFF
Confidence 1 — Organism
Curated By Intermediate

Target

HFF (CHEMBL614071)
Type CELL-LINE
Organism Homo sapiens

Publication

Benzimidazole ribonucleosides: Observation of an unexpected nitration when performing non-aqueous diazotizations with t-butyl nitrite
Devivar RV, Drach JC, Townsend LB
Bioorg Med Chem Lett (1992) 2 : 1105 -1110
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 4.28 4.62

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL375530 DICHLORORIBOBENZIMIDAZOLE 1 4.62
CHEMBL603513 1 4.50
CHEMBL608658 1 4.00
CHEMBL608318 1 4.00
CHEMBL605800 1 -
CHEMBL182 GANCICLOVIR 4.0 1 -
CHEMBL605799 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL375530 DICHLORORIBOBENZIMIDAZOLE IC50 = 24000.0 nM 4.62
CHEMBL603513 IC50 = 32000.0 nM 4.50
CHEMBL608658 IC50 = 100000.0 nM 4.00
CHEMBL608318 IC50 = 100000.0 nM 4.00
CHEMBL605800 IC50 = 127000.0 nM -
CHEMBL182 GANCICLOVIR IC50 > 100000.0 nM -
CHEMBL605799 IC50 > 100000.0 nM -