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Compound Detail

CHEMBL608658

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O=[N+]([O-])c1c(Cl)c(Cl)cc2c1nc(O)n2C1O[C@H](CO)[C@@H](O)[C@H]1O

Basic Information

ChEMBL ID CHEMBL608658
Phase Preclinical
Structure Type MOL
InChI Key VJIJPZLRHFYQRV-ZBCCYFLUSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
6
Publications
0
Known Names

Molecular Properties

380.1
MW (Da)
0.57
ALogP
9
HBA
4
HBD
151.1
PSA (Ų)
0.45
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C12H11Cl2N3O7
MW 380.14
Aromatic Rings 2
Heavy Atoms 24
NP-Likeness 0.20

Activity Summary

IC50 2 meas. best 4.0

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
HFF
CHEMBL614071
IC50 4.0 4.0 100000.0 2

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
HFF IC50 = 100000.0 nM 4.0 Compound was evaluated for the visual cytotoxicity scored on HFF cells at time o... 7562945
HFF IC50 = 100000.0 nM 4.0 Cytotoxicity against human foreskin fibroblasts (HFF) cells -

Literature References

PubMed DOI Target Context # Activities
7562945 10.1021/jm00020a025 Human betaherpesvirus 5 1
7562945 10.1021/jm00020a025 Human alphaherpesvirus 1 1
7562945 10.1021/jm00020a025 HFF 1
- 10.1016/S0960-894X(00)80628-9 Human betaherpesvirus 5 1
- 10.1016/S0960-894X(00)80628-9 Human alphaherpesvirus 1 1
- 10.1016/S0960-894X(00)80628-9 HFF 1

Data from ChEMBL 36 via Core Engine