Assay Detail
Functional
CHEMBL697148
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Compound was tested for the antiviral activity against Human Rhinovirus -14(HRV-14) in HeLa cells
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HeLa |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Design, synthesis, and evaluation of nonpeptidic inhibitors of human rhinovirus 3C protease.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 12 | 4.53 | 5.20 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL150011 | — | — | 1 | 5.20 |
| CHEMBL348660 | — | — | 1 | 4.85 |
| CHEMBL64582 | — | — | 1 | 4.25 |
| CHEMBL148483 | — | — | 1 | 4.18 |
| CHEMBL64413 | — | — | 1 | 4.15 |
| CHEMBL146403 | — | — | 1 | - |
| CHEMBL149950 | — | — | 1 | - |
| CHEMBL149822 | — | — | 1 | - |
| CHEMBL149227 | — | — | 1 | - |
| CHEMBL149556 | — | — | 1 | - |
| CHEMBL145833 | — | — | 1 | - |
| CHEMBL358279 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL150011 | — | EC50 | = | 6300.0 | nM | 5.20 |
| CHEMBL348660 | — | EC50 | = | 14100.0 | nM | 4.85 |
| CHEMBL64582 | — | EC50 | = | 56000.0 | nM | 4.25 |
| CHEMBL148483 | — | EC50 | = | 66000.0 | nM | 4.18 |
| CHEMBL64413 | — | EC50 | = | 71000.0 | nM | 4.15 |
| CHEMBL146403 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL149950 | — | EC50 | > | 5600.0 | nM | - |
| CHEMBL149822 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL149227 | — | EC50 | > | 7100.0 | nM | - |
| CHEMBL149556 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL145833 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL358279 | — | EC50 | > | 10000.0 | nM | - |