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Assay Detail

CHEMBL697551

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Functional
Inhibitory concentration against human cytomegalovirus (HCMV) in plaque reduction assay
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human betaherpesvirus 5
Confidence 1 — Organism
Curated By Expert

Target

Human betaherpesvirus 5 (CHEMBL371)
Type ORGANISM
Organism Human betaherpesvirus 5

Publication

Synthesis and antiviral activity of certain 4- and 4,5-disubstituted 7-[(2-hydroxyethoxy)methyl]pyrrolo[2,3-d]pyrimidines.
Pudlo JS, Saxena NK, Nassiri MR, Turk SR, Drach JC, Townsend LB.
J Med Chem (1988) 31 : 2086 -2092
PubMed 2846837 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 11 5.35 6.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL99203 IODOTUBERCIDIN 1 6.40
CHEMBL62099 1 6.30
CHEMBL3126906 1 5.92
CHEMBL1688967 IMMUNICILLIN H 1 5.46
CHEMBL610074 1 5.40
CHEMBL98933 1 5.36
CHEMBL403715 1 5.00
CHEMBL612156 1 4.64
CHEMBL610644 1 4.54
CHEMBL328824 1 4.51
CHEMBL610642 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL99203 IODOTUBERCIDIN IC50 = 400.0 nM 6.40
CHEMBL62099 IC50 = 500.0 nM 6.30
CHEMBL3126906 IC50 = 1200.0 nM 5.92
CHEMBL1688967 IMMUNICILLIN H IC50 = 3500.0 nM 5.46
CHEMBL610074 IC50 = 4000.0 nM 5.40
CHEMBL98933 IC50 = 4400.0 nM 5.36
CHEMBL403715 IC50 = 10000.0 nM 5.00
CHEMBL612156 IC50 = 23000.0 nM 4.64
CHEMBL610644 IC50 = 29000.0 nM 4.54
CHEMBL328824 IC50 = 31000.0 nM 4.51
CHEMBL610642 IC50 > 100000.0 nM -