Assay Detail
Binding
CHEMBL699440
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory concentration of compound against strand transfer of of HIV-2 integrase
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Human immunodeficiency virus 2 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Human immunodeficiency virus type 2 integrase (CHEMBL3463) ↗| Type | SINGLE PROTEIN |
| Organism | Human immunodeficiency virus 2 |
Publication
Depsides and depsidones as inhibitors of HIV-1 integrase: discovery of novel inhibitors through 3D database searching.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.82 | 5.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL175266 | — | — | 1 | 5.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL175266 | — | IC50 | = | 1500.0 | nM | 5.82 |