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Assay Detail

CHEMBL699693

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity against mouse Inducible nitric oxide synthase (iNOS)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Nitric oxide synthase, inducible (CHEMBL3464)
Type SINGLE PROTEIN
Organism Mus musculus

Publication

Synthesis and evaluation of two positron-labeled nitric oxide synthase inhibitors, S-[11C]methylisothiourea and S-(2-[18F]fluoroethyl)isothiourea, as potential positron emission tomography tracers.
Zhang J, McCarthy TJ, Moore WM, Currie MG, Welch MJ.
J Med Chem (1996) 39 : 5110 -5118
PubMed 8978842 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 8.28 8.28

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL321691 ETHYLISOTHIOUREA 1 8.28

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL321691 ETHYLISOTHIOUREA Ki = 5.2 nM 8.28