Assay Detail
Functional
CHEMBL699999
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonistic activity was determined by measuring the ability to inhibit superoxide production (stimulated by fMLF) using human neutrophils
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
N-terminus urea-substituted chemotactic peptides: new potent agonists and antagonists toward the neutrophil fMLF receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 15 | 6.06 | 7.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL7486 | — | — | 1 | 7.70 |
| CHEMBL6450 | — | — | 1 | 7.00 |
| CHEMBL415296 | — | — | 1 | 6.52 |
| CHEMBL162488 | — | — | 1 | 6.30 |
| CHEMBL7122 | — | — | 1 | 6.30 |
| CHEMBL7363 | — | — | 1 | 6.22 |
| CHEMBL7226 | — | — | 1 | 6.22 |
| CHEMBL6997 | — | — | 1 | 5.80 |
| CHEMBL6779 | — | — | 1 | 5.70 |
| CHEMBL7181 | — | — | 1 | 5.70 |
| CHEMBL415299 | — | — | 1 | 5.70 |
| CHEMBL266448 | — | — | 1 | 5.52 |
| CHEMBL7214 | — | — | 1 | 5.52 |
| CHEMBL268823 | — | — | 1 | 5.40 |
| CHEMBL7034 | — | — | 1 | 5.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL7486 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL6450 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL415296 | — | IC50 | = | 300.0 | nM | 6.52 |
| CHEMBL162488 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL7122 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL7363 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL7226 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL6997 | — | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL6779 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL7181 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL415299 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL266448 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL7214 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL268823 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL7034 | — | IC50 | = | 5000.0 | nM | 5.30 |