Assay Detail
Functional
CHEMBL700458
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Evaluated for inhibition of 4 uM ADP-induced human platelet aggregation
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Molecular design of novel PGI2 agonists without PG skeleton. I
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.82 | 5.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL10742 | — | — | 1 | 5.96 |
| CHEMBL10470 | — | — | 1 | 5.68 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL10742 | — | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL10470 | — | IC50 | = | 2100.0 | nM | 5.68 |