Assay Detail
Functional
CHEMBL700482
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The compound was tested ex vivo at a dose of 0.08 mmol/kg for ADP induced platelet aggregation in guinea pig
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Inhibitors of blood platelet aggregation. Effects of some 1,2-benzisothiazol-3-ones on platelet responsiveness to adenosine diphosphate and collagen.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.49 | 4.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL417351 | — | — | 1 | 4.77 |
| CHEMBL298460 | — | — | 1 | 4.20 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL417351 | — | IC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL298460 | — | IC50 | = | 63000.0 | nM | 4.20 |