Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL700623

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against uninfected human foreskin fibroblast(HFF cells)
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HFF
Confidence 1 — Organism
Curated By Expert

Target

HFF (CHEMBL614071)
Type CELL-LINE
Organism Homo sapiens

Publication

Synthesis and antiviral activity of certain 4- and 4,5-disubstituted 7-[(2-hydroxyethoxy)methyl]pyrrolo[2,3-d]pyrimidines.
Pudlo JS, Saxena NK, Nassiri MR, Turk SR, Drach JC, Townsend LB.
J Med Chem (1988) 31 : 2086 -2092
PubMed 2846837 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 11 5.07 5.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL610074 1 5.70
CHEMBL99203 IODOTUBERCIDIN 1 5.70
CHEMBL3126906 1 5.70
CHEMBL62099 1 5.35
CHEMBL98933 1 5.00
CHEMBL1688967 IMMUNICILLIN H 1 5.00
CHEMBL328824 1 4.89
CHEMBL612156 1 4.51
CHEMBL610644 1 4.51
CHEMBL403715 1 4.34
CHEMBL610642 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL610074 IC50 = 2000.0 nM 5.70
CHEMBL99203 IODOTUBERCIDIN IC50 = 2000.0 nM 5.70
CHEMBL3126906 IC50 = 2000.0 nM 5.70
CHEMBL62099 IC50 = 4500.0 nM 5.35
CHEMBL98933 IC50 = 10000.0 nM 5.00
CHEMBL1688967 IMMUNICILLIN H IC50 = 10000.0 nM 5.00
CHEMBL328824 IC50 = 13000.0 nM 4.89
CHEMBL612156 IC50 = 31000.0 nM 4.51
CHEMBL610644 IC50 = 31000.0 nM 4.51
CHEMBL403715 IC50 = 46000.0 nM 4.34
CHEMBL610642 IC50 > 100000.0 nM -