Assay Detail
Functional
CHEMBL701918
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of LPS-induced PGE-2 production in the human whole blood.
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Tissue | Blood |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
1,2-Diarylpyrroles as potent and selective inhibitors of cyclooxygenase-2.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.36 | 5.36 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL43755 | — | — | 1 | 5.36 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL43755 | — | IC50 | = | 4400.0 | nM | 5.36 |