Assay Detail
Functional
CHEMBL702046
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In vitro ability to inhibit arachidonic acid induced platelet aggregation (AAIPA)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Conformationally-restricted analogs of TXA2 antagonist SQ 33,961: Receptor binding conformation of the carboxyl sidechain
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 7.23 | 8.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL31765 | — | — | 1 | 8.70 |
| CHEMBL343679 | — | — | 1 | 8.10 |
| CHEMBL357372 | — | — | 1 | 4.90 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL31765 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL343679 | — | IC50 | = | 8.0 | nM | 8.10 |
| CHEMBL357372 | — | IC50 | = | 12700.0 | nM | 4.90 |