Assay Detail
Binding
CHEMBL709304
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Compound was tested for inhibitory activity against human neutrophil LTB4 receptor binding
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Modulators of leukotriene biosynthesis and receptor activation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 8.38 | 8.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL419948 | — | — | 1 | 8.89 |
| CHEMBL328492 | — | — | 1 | 8.82 |
| CHEMBL88337 | — | — | 1 | 8.40 |
| CHEMBL90788 | — | — | 1 | 7.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL419948 | — | IC50 | = | 1.3 | nM | 8.89 |
| CHEMBL328492 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL88337 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL90788 | — | IC50 | = | 39.6 | nM | 7.40 |