Assay Detail
Binding
CHEMBL709863
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Compound was tested for inhibitory activity against human neutrophil LTB4 receptor binding
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Modulators of leukotriene biosynthesis and receptor activation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 8.45 | 9.33 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL292782 | — | — | 1 | 9.33 |
| CHEMBL422420 | — | — | 1 | 8.43 |
| CHEMBL329123 | ETALOCIB | 2.0 | 1 | 7.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL292782 | — | Ki | = | 0.47 | nM | 9.33 |
| CHEMBL422420 | — | Ki | = | 3.7 | nM | 8.43 |
| CHEMBL329123 | ETALOCIB | Ki | = | 25.0 | nM | 7.60 |