Assay Detail
Functional
CHEMBL710019
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Effective concentration was measured against frog skin(MCR) cells at 10 e-4 10 e-12 M Concentration.
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | frog |
| Cell Type | MCR |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Discovery of prototype peptidomimetic agonists at the human melanocortin receptors MC1R and MC4R.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 5.17 | 5.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL65339 | — | — | 1 | 5.82 |
| CHEMBL432895 | — | — | 1 | 4.52 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL65339 | — | EC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL432895 | — | EC50 | = | 30000.0 | nM | 4.52 |