Assay Detail
Functional
CHEMBL710306
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of growth in uninfected MT-4 cells in MTM assay
29
Total Activities
29
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MT4 |
| Confidence | 1 — Organism |
| Curated By | Expert |
Publication
Synthesis and anti-HIV-1 activity of a series of imidazo[1,5-b]pyridazines.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 29 | 4.58 | 4.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL124248 | — | — | 1 | 4.60 |
| CHEMBL124271 | — | — | 1 | 4.60 |
| CHEMBL123514 | — | — | 1 | 4.60 |
| CHEMBL125205 | — | — | 1 | 4.60 |
| CHEMBL435017 | — | — | 1 | 4.58 |
| CHEMBL125532 | — | — | 1 | 4.58 |
| CHEMBL125446 | — | — | 1 | 4.58 |
| CHEMBL338099 | — | — | 1 | 4.58 |
| CHEMBL338302 | — | — | 1 | 4.58 |
| CHEMBL434441 | — | — | 1 | 4.58 |
| CHEMBL121820 | — | — | 1 | 4.58 |
| CHEMBL341512 | — | — | 1 | 4.57 |
| CHEMBL1203237 | — | — | 1 | 4.57 |
| CHEMBL332351 | — | — | 1 | 4.55 |
| CHEMBL338823 | — | — | 1 | 4.52 |
| CHEMBL341238 | — | — | 1 | - |
| CHEMBL127427 | — | — | 1 | - |
| CHEMBL1203236 | — | — | 1 | - |
| CHEMBL435216 | — | — | 1 | - |
| CHEMBL338415 | — | — | 1 | - |
| CHEMBL126811 | — | — | 1 | - |
| CHEMBL338339 | — | — | 1 | - |
| CHEMBL123202 | — | — | 1 | - |
| CHEMBL126216 | — | — | 1 | - |
| CHEMBL341350 | — | — | 1 | - |
| CHEMBL340248 | — | — | 1 | - |
| CHEMBL124246 | — | — | 1 | - |
| CHEMBL125084 | — | — | 1 | - |
| CHEMBL123839 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL124248 | — | IC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL124271 | — | IC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL123514 | — | IC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL125205 | — | IC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL435017 | — | IC50 | = | 26000.0 | nM | 4.58 |
| CHEMBL125532 | — | IC50 | = | 26000.0 | nM | 4.58 |
| CHEMBL125446 | — | IC50 | = | 26000.0 | nM | 4.58 |
| CHEMBL338099 | — | IC50 | = | 26000.0 | nM | 4.58 |
| CHEMBL338302 | — | IC50 | = | 26000.0 | nM | 4.58 |
| CHEMBL434441 | — | IC50 | = | 26000.0 | nM | 4.58 |
| CHEMBL121820 | — | IC50 | = | 26000.0 | nM | 4.58 |
| CHEMBL341512 | — | IC50 | = | 27000.0 | nM | 4.57 |
| CHEMBL1203237 | — | IC50 | = | 27000.0 | nM | 4.57 |
| CHEMBL332351 | — | IC50 | = | 28000.0 | nM | 4.55 |
| CHEMBL338823 | — | IC50 | = | 30000.0 | nM | 4.52 |
| CHEMBL341238 | — | IC50 | = | 250000.0 | nM | - |
| CHEMBL127427 | — | IC50 | = | 260000.0 | nM | - |
| CHEMBL1203236 | — | IC50 | = | 250000.0 | nM | - |
| CHEMBL435216 | — | IC50 | = | 290000.0 | nM | - |
| CHEMBL338415 | — | IC50 | = | 260000.0 | nM | - |
| CHEMBL126811 | — | IC50 | = | 250000.0 | nM | - |
| CHEMBL338339 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL123202 | — | IC50 | = | 260000.0 | nM | - |
| CHEMBL126216 | — | IC50 | = | 260000.0 | nM | - |
| CHEMBL341350 | — | IC50 | < | 30.0 | nM | - |
| CHEMBL340248 | — | IC50 | = | 280000.0 | nM | - |
| CHEMBL124246 | — | IC50 | = | 250000.0 | nM | - |
| CHEMBL125084 | — | IC50 | = | 250000.0 | nM | - |
| CHEMBL123839 | — | IC50 | = | 250000.0 | nM | - |