Assay Detail
Functional
CHEMBL712362
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Tested for inhibition of cytopathic effect of HIV-2ROD in MT-4 cells
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MT4 |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Anti-HIV activity of a series of cosalane amino acid conjugates.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 10 | 4.55 | 5.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3138187 | — | — | 1 | 5.40 |
| CHEMBL3138374 | — | — | 1 | 4.14 |
| CHEMBL3138360 | — | — | 1 | 4.12 |
| CHEMBL3137850 | — | — | 1 | - |
| CHEMBL3138117 | — | — | 1 | - |
| CHEMBL3138122 | — | — | 1 | - |
| CHEMBL3138094 | — | — | 1 | - |
| CHEMBL3137855 | — | — | 1 | - |
| CHEMBL3137853 | — | — | 1 | - |
| CHEMBL3137848 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3138187 | — | EC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL3138374 | — | EC50 | = | 71600.0 | nM | 4.14 |
| CHEMBL3138360 | — | EC50 | = | 75200.0 | nM | 4.12 |
| CHEMBL3137850 | — | EC50 | > | 125000.0 | nM | - |
| CHEMBL3138117 | — | EC50 | = | 122000.0 | nM | - |
| CHEMBL3138122 | — | EC50 | > | 62000.0 | nM | - |
| CHEMBL3138094 | — | EC50 | > | 125000.0 | nM | - |
| CHEMBL3137855 | — | EC50 | > | 125000.0 | nM | - |
| CHEMBL3137853 | — | EC50 | = | 120000.0 | nM | - |
| CHEMBL3137848 | — | EC50 | > | 125000.0 | nM | - |