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Assay Detail

CHEMBL713550

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Concentration of compound required to reduce MT-4 cell viability by 50%
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MT4
Confidence 1 — Organism
Curated By Intermediate

Target

MT4 (CHEMBL388)
Type CELL-LINE
Organism Homo sapiens

Publication

Chicoric acid analogues as HIV-1 integrase inhibitors.
Lin Z, Neamati N, Zhao H, Kiryu Y, Turpin JA, Aberham C, Strebel K, Kohn K, Witvrouw M, Pannecouque C, Debyser Z, De Clercq E, Rice WG, Pommier Y, Burke TR.
J Med Chem (1999) 42 : 1401 -1414
PubMed 10212126 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 4.26 4.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL29660 CHICORIC ACID 1 4.40
CHEMBL282731 CICHORIC ACID 1 4.35
CHEMBL29369 1 4.33
CHEMBL30455 1 4.22
CHEMBL129 ZIDOVUDINE 4.0 1 4.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL29660 CHICORIC ACID IC50 = 39700.0 nM 4.40
CHEMBL282731 CICHORIC ACID IC50 = 45000.0 nM 4.35
CHEMBL29369 IC50 = 47100.0 nM 4.33
CHEMBL30455 IC50 = 60000.0 nM 4.22
CHEMBL129 ZIDOVUDINE IC50 = 100000.0 nM 4.00