Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL714334

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Anti-HIV-1 activity against Y181C strain, in MT-4 cells by the MTT method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MT4
Confidence 1 — Organism
Curated By Intermediate

Target

MT4 (CHEMBL388)
Type CELL-LINE
Organism Homo sapiens

Publication

3-iodo-4-phenoxypyridinones (IOPY's), a new family of highly potent non-nucleoside inhibitors of HIV-1 reverse transcriptase.
Benjahad A, Guillemont J, Andries K, Nguyen CH, Grierson DS.
Bioorg Med Chem Lett (2003) 13 : 4309 -4312
PubMed 14643315 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.70 7.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL233664 1 7.70

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL233664 IC50 = 20.0 nM 7.70