Assay Detail
Binding
CHEMBL714606
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Effective concentration required for the biological activity against human Melanocortin 4 receptor
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Peptide science: exploring the use of chemical principles and interdisciplinary collaboration for understanding life processes.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3 | 10.23 | 10.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL441738 | AFAMELANOTIDE | 4.0 | 1 | 10.77 |
| CHEMBL430239 | MELATONAN | — | 1 | 10.24 |
| CHEMBL214332 | INTERMEDINE | 2.0 | 1 | 9.68 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL441738 | AFAMELANOTIDE | EC50 | = | 0.017 | nM | 10.77 |
| CHEMBL430239 | MELATONAN | EC50 | = | 0.057 | nM | 10.24 |
| CHEMBL214332 | INTERMEDINE | EC50 | = | 0.21 | nM | 9.68 |