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Assay Detail

CHEMBL715876

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Binding
Binding affinity towards melatonin receptor in Chicken brain Experiment 2
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 4 — Cell-line / Tissue
Curated By Autocuration

Target

Melatonin receptor (CHEMBL2095154)
Type PROTEIN FAMILY
Organism Gallus gallus

Publication

Mapping the melatonin receptor. 4. Comparison of the binding affinities of a series of substituted phenylalkyl amides.
Garratt PJ, Travard S, Vonhoff S, Tsotinis A, Sugden D.
J Med Chem (1996) 39 : 1797 -1805
PubMed 8627603 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 2 6.60 6.60

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL53722 1 6.60
CHEMBL53721 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL53722 Ki = 253.0 nM 6.60
CHEMBL53721 Ki > 1000.0 nM -