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Assay Detail

CHEMBL717596

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
pA2 against human melanocortin receptor, human Melanocortin 4 receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Melanocortin receptor 4 (CHEMBL259)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Peptide science: exploring the use of chemical principles and interdisciplinary collaboration for understanding life processes.
Hruby VJ.
J Med Chem (2003) 46 : 4215 -4231
PubMed 13678399 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 2 9.50 9.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL440801 1 9.70
CHEMBL2096742 1 9.30

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL440801 Kd = 0.1995 nM 9.70
CHEMBL2096742 Kd = 0.5012 nM 9.30