Assay Detail
Functional
CHEMBL732613
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Inhibition of p38 MAP kinase related interleukin (IL1-beta (cytokine) release from human whole blood
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Tissue | Blood |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
From imidazoles to pyrimidines: new inhibitors of cytokine release.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 10 | 5.05 | 5.56 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL111456 | — | — | 1 | 5.56 |
| CHEMBL358814 | — | — | 1 | 5.40 |
| CHEMBL143370 | — | — | 1 | 5.39 |
| CHEMBL313417 | — | — | 1 | 4.57 |
| CHEMBL92723 | — | — | 1 | 4.34 |
| CHEMBL92070 | — | — | 1 | - |
| CHEMBL94086 | — | — | 1 | - |
| CHEMBL92724 | — | — | 1 | - |
| CHEMBL93574 | — | — | 1 | - |
| CHEMBL93914 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL111456 | — | IC50 | = | 2780.0 | nM | 5.56 |
| CHEMBL358814 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL143370 | — | IC50 | = | 4100.0 | nM | 5.39 |
| CHEMBL313417 | — | IC50 | = | 27000.0 | nM | 4.57 |
| CHEMBL92723 | — | IC50 | = | 45500.0 | nM | 4.34 |
| CHEMBL92070 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL94086 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL92724 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL93574 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL93914 | — | IC50 | > | 100000.0 | nM | - |