Assay Detail
Binding
CHEMBL732792
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In vitro binding affinity towards human motilin receptor
12
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Discovery of a potent and novel motilin agonist.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 12 | 7.50 | 9.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL297494 | — | — | 2 | 9.15 |
| CHEMBL296748 | — | — | 1 | 8.70 |
| CHEMBL298224 | — | — | 1 | 8.57 |
| CHEMBL2372767 | MOTILIN | — | 1 | 8.51 |
| CHEMBL1628277 | — | — | 1 | 8.47 |
| CHEMBL45905 | — | — | 3 | 5.39 |
| CHEMBL532 | ERYTHROMYCIN | 4.0 | 1 | 4.43 |
| CHEMBL46272 | — | — | 1 | - |
| CHEMBL33827 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL297494 | — | Ki | = | 0.7 | nM | 9.15 |
| CHEMBL297494 | — | Ki | = | 1.0 | nM | 9.00 |
| CHEMBL296748 | — | Ki | = | 2.0 | nM | 8.70 |
| CHEMBL298224 | — | Ki | = | 2.7 | nM | 8.57 |
| CHEMBL2372767 | MOTILIN | Ki | = | 3.1 | nM | 8.51 |
| CHEMBL1628277 | — | Ki | = | 3.4 | nM | 8.47 |
| CHEMBL45905 | — | Ki | = | 4100.0 | nM | 5.39 |
| CHEMBL45905 | — | Ki | = | 5800.0 | nM | 5.24 |
| CHEMBL532 | ERYTHROMYCIN | Ki | = | 37000.0 | nM | 4.43 |
| CHEMBL46272 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL33827 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL45905 | — | Ki | > | 10000.0 | nM | - |