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Assay Detail

CHEMBL746596

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibition of electrically evoked contractions in mouse vas deferens
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Confidence 9 — Direct single protein target
Curated By Expert

Target

Delta-type opioid receptor (CHEMBL3222)
Type SINGLE PROTEIN
Organism Mus musculus

Publication

Conformationally restricted deltorphin analogues.
Schiller PW, Weltrowska G, Nguyen TM, Wilkes BC, Chung NN, Lemieux C.
J Med Chem (1992) 35 : 3956 -3961
PubMed 1331451 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 9.15 9.15

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL436590 1 9.15

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL436590 IC50 = 0.712 nM 9.15